Compile Data Set for Download or QSAR
maximum 50k data
Found 28 of ic50 data for polymerid = 4426
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
Affinity DataIC50:  0.0160nMAssay Description:Inhibition of cAMP dependent Protein kinase A of rabbit Skeletal Muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM36603(4'',6''-Dideoxybalanol, 6)
Affinity DataKi:  3.40nM ΔG°:  -11.7kcal/mole IC50:  5.5nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM36604(5'-Deoxybalanol, 7)
Affinity DataKi:  3.5nM ΔG°:  -11.7kcal/mole IC50:  5.70nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM3207(10''-Deoxybalanol, 4 | 2-{[2,6-dihydroxy-4-({[(3R,...)
Affinity DataKi:  3.90nM ΔG°:  -11.7kcal/mole IC50:  6.30nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
Affinity DataIC50: >10nMAssay Description:Inhibition of cAMP dependent Protein kinase A of rabbit Skeletal Muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM36602(14''-Decarboxybalanol hydrochloride, 5)
Affinity DataKi:  11nM ΔG°:  -11.0kcal/mole IC50:  18nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM2672(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM2583(3,4-Bis(3-indolyl)-1H-pyrrole-2,5-dione | 3,4-bis(...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040920(5,6-Bis-p-tolylamino-isoindole-1,3-dione | CHEMBL7...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040914(5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040926(4,5-Bis-phenylamino-phthalic acid dimethyl ester |...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040919(5,6-Bis-(biphenyl-4-ylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040929(4,5-dianilinophthalimide | 5,6-bis(phenylamino)-1H...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040915(5,6-Bis-(4-iodo-phenylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040927(CHEMBL268441 | N-(1,3-Dioxo-6-phenylamino-2,3-dihy...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040931(4,5-Bis-(4-fluoro-phenylamino)-phthalic acid dimet...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040913(1,4-Diphenyl-1,2,3,4-tetrahydro-pyrrolo[3,4-g]quin...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040928(4-[6-(4-cyanoanilino)-1,3-dioxo-2,3-dihydro-1H-5-i...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040923(2-Methyl-5,6-bis-phenylamino-isoindole-1,3-dione |...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040916(5,6-Bis-(4-hydroxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040912(5,6-Bis-cyclohexylamino-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040922(2-Phenyl-5,6-bis-phenylamino-isoindole-1,3-dione |...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040921(5,6-Bis-(4-diethylamino-phenylamino)-isoindole-1,3...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040925(5,6-Bis-(4-methoxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040924(5,6-Bis-phenylsulfanyl-isoindole-1,3-dione | CHEMB...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040918(5,6-Bis-(methyl-phenyl-amino)-isoindole-1,3-dione ...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed